We established a kinase profiling platform with 520 human kinase domains. This platform allows examining inhibitor potency and specificity in cellular lysates, providing an advantage over readily-available biochemical solutions.

1. We offer a complete scan of the kinome (520 K_D values), provided the compound to test can be labeled with a fluorophore. Kinetics are also feasible. Please contact us to discuss your needs.

2. Alternatively, we offer readily-available assays for 288 kinase domains, enabling K_I determination of label-free test compounds. Kinetics are also feasible. Please contact us to discuss your needs.